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Purpose
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Gedatolisib (PF-05212384, PKI-587) is a highly potent dual inhibitor of PI3Kα, PI3Kγ and mTOR with IC50 of 0.4 nM, 5.4 nM and 1.6 nM in cell-free assays, respectively. Phase 2.
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Characteristics
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Target: PI3K inhibitor, mTOR inhibitor
Receptor: PI3Kα, mTOR, PI3Kγ
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Purification
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All the products are sent with COA, HPLC and NMR inspection report to guarantee the quality.
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Purity
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98?%
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Formula
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C32H41N9O4
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Solubility
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Soluble in DMSO
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