產品詳情
簡單介紹:
[Boc-Asp(Obzl)-Lys(z)-OtBu],Reversin121
詳情介紹:
Purity | 98 % |
Background | Selective high affinity inhibitor of Pgp (MDR1). IC50 of Pgp-dependent Calcein-AM extrusion = 0.3 μM, IC50 of MRP1-dependent Calcein-AM extrusion = 1.8 μM, EC50 for Pgp ATPase activity = 0.2 μM. |
Molecular Weight | 642 Da |
Comment |
Formula: C34H47N3O9 |
Restrictions | For Research Use only |
Format | Powder |
Reconstitution | Soluble in DMSO. Melting Point: 80-90°C |
Storage | -20 °C |