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  • 產(chǎn)品名稱:AKR1C3InhibitorIII

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  • 產(chǎn)品廠商:Biovision
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簡單介紹:
AKR1C3InhibitorIII
詳情介紹:
Purpose A highly potent and selective inhibitor of the type 5 17-beta-hydroxysteroid dehydrogenase AKR1C3
Characteristics A highly potent and selective inhibitor of the type 5 17-beta-hydroxysteroid dehydrogenase AKR1C3 (IC50= 88 nM). Displays > 100-fold selectivity against AKR1C1, AKR1C2 and AKR1C4. Does not display any COX (cyclooxygenase) inhibition at 10 μM in whole blood assay.
Purity ≥ 98?% by HPLC
Chemical Name 4-(4-Chlorophenyl)piperazin-1-yl)(morpholino)methanone
Formula C??H??ClN?O?
Permeability Cell-permeable
Solubility DMSO
Molecular Weight 309.79 g/mol
Restrictions For Research Use only
Format Solid
Handling Advice Protect from air and light
Storage -20 °C
Expiry Date 36 months
Supplier Images
 image for AKR1C3 Inhibitor III (ABIN1685859) AKR1C3 Inhibitor III
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